mometasone furoate
Ligand Summary
A pregnadienediol derivative ANTI-ALLERGIC AGENT and ANTI-INFLAMMATORY AGENT that is used in the management of ASTHMA and ALLERGIC RHINITIS. It is also used as a topical treatment for skin disorders.
UNII: 04201GDN4R
PubChem: 441336
ChEMBL: CHEMBL1161
DrugCentral: 1832
LyCHI: LQ9FLU1BPCR8
Target Activities
NR3C1
Glucocorticoid receptor
2 Activities
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1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Ki | 9.15 | J Med Chem, (2019) 62:22:10005 | ||||
Ki | 9.15 | AGONIST | ||||
PGR
Progesterone receptor
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 10.1 | J. Med. Chem., (2004) 47:13:3381 | ||||
SLCO1B3
Solute carrier organic anion transporter family member 1B3
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Ki | 6.06 | Mol. Pharmacol., (2013) 83:6:1257 | ||||