betahistine
Ligand Summary
A histamine analog and H1 receptor agonist that serves as a vasodilator. It is used in MENIERE DISEASE and in vascular headaches but may exacerbate bronchial asthma and peptic ulcers.
UNII: X32KK4201D
ChEMBL: CHEMBL4298035
DrugCentral: 346
LyCHI: JSTBVXS1B5JX
Target Activities
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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EC50 | INVERSE AGONIST | |||||