Pharos: Illuminating the Druggable Genome

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Ligand Summary

Ligand Structure

chemical structure image

Synonyms & Links

NCATS Inxight: Drugs: 17759043

Name: 4-bromo-3-carboxymethoxy-5-[3-(3,3,5,5-tetramethylcyclohexylamino)phenyl]thiophene-2-carboxylic acid

PubChem: 17759043

ChEMBL: CHEMBL243942

LyCHI: RQ76K2DFXRAP

Target Activities

Items per page:

10

1 – 2 of 2

PTPN1

Tchem

Tyrosine-protein phosphatase non-receptor type 1

2 Activities

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1 – 2 of 2

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
Ki	7.44		J. Med. Chem., (2007) 50:19:4681	17705360

Ki	7.58		J. Med. Chem., (2009) 52:21:6649	19810703

PTPN2

Tchem

Tyrosine-protein phosphatase non-receptor type 2

2 Activities

Items per page:

1 – 2 of 2

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
Ki	7.44		J. Med. Chem., (2009) 52:21:6649	19810703

Ki	7.58		J. Med. Chem., (2007) 50:19:4681	17705360