CHEMBL4072812
Ligand Summary
Name: rac-6-(4-Methylpiperazin-1-yl)-2-(1,3,6-trimethyl-2-oxo-2,3-dihydro-1H-benzimidazol-5-yl)-1H-benzo[de]isoquinoline-1,3(2H)-dione
PubChem: 130471724
ChEMBL: CHEMBL4072812
LyCHI: BLH2D5P219VW
Target Activities
BRPF1
Peregrin
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 6 | J Med Chem, (2017) 60:9:4002 | ||||
BRD1
Bromodomain-containing protein 1
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 7.03 | J Med Chem, (2017) 60:9:4002 | ||||
TAF1
Transcription initiation factor TFIID subunit 1
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 8.4 | J Med Chem, (2017) 60:9:4002 | ||||