Pharos : Ligand Details - BDL2TN46DL4B

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Ligand Summary

Ligand Structure

Rendered image for the query structure

Synonyms & Links

Name: 8-(((3R,4R)-3-((1,1-Dioxidotetrahydro-2H-thiopyran-4-yl)-methoxy)-1-methylpiperidin-4-yl)amino)-3-methyl-5-(5-methylpyridin-3-yl)-1,7-naphthyridin-2(1H)-one

PubChem: 122181572

ChEMBL: CHEMBL3590408

LyCHI: BDL2TN46DL4B

Target Activities

Explore Associated and Predicted Targets

ATAD2

Tchem

ATPase family AAA domain-containing protein 2

8 Activities

Items per page:

1 – 8 of 8

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
Ki	7.7		J. Med. Chem., (2015) 58:15:6151	26230603

Ki	7.7		J. Med. Chem., (2015) 58:15:6151	26230603

Kd	7.2		J. Med. Chem., (2015) 58:15:6151	26230603

IC50	7		J. Med. Chem., (2015) 58:15:6151	26230603

Kd	6.7		J. Med. Chem., (2015) 58:15:6151	26230603

Kd	6.7		J. Med. Chem., (2015) 58:15:6151	26230603

IC50	6.6		J. Med. Chem., (2015) 58:15:6151	26230603

IC50	6.5		J. Med. Chem., (2015) 58:15:6151	26230603

ATAD2B

Tchem

ATPase family AAA domain-containing protein 2B

2 Activities

Items per page:

1 – 2 of 2

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
Ki	7.4		J. Med. Chem., (2015) 58:15:6151	26230603

Kd	7		J. Med. Chem., (2015) 58:15:6151	26230603

BRD1

Tchem

Bromodomain-containing protein 1

1 Activities

Items per page:

1 – 1 of 1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
Ki	6.4		J. Med. Chem., (2015) 58:15:6151	26230603

CECR2

Tchem

Cat eye syndrome critical region protein 2

1 Activities

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1 – 1 of 1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
Ki	6.1		J. Med. Chem., (2015) 58:15:6151	26230603

TAF1L

Tchem

Transcription initiation factor TFIID subunit 1-like

1 Activities

Items per page:

1 – 1 of 1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
Ki	6.9		J. Med. Chem., (2015) 58:15:6151	26230603

BRPF3

Tchem

Bromodomain and PHD finger-containing protein 3

1 Activities

Items per page:

1 – 1 of 1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
Ki	6.1		J. Med. Chem., (2015) 58:15:6151	26230603