doxepin
Ligand Summary
A dibenzoxepin tricyclic compound. It displays a range of pharmacological actions including maintaining adrenergic innervation. Its mechanism of action is not fully understood, but it appears to block reuptake of monoaminergic neurotransmitters into presynaptic terminals. It also possesses anticholinergic activity and modulates antagonism of histamine H(1)- and H(2)-receptors.
UNII: 851NLB57HQ
PubChem: 3158
ChEMBL: CHEMBL1628227
DrugCentral: 956
LyCHI: VP4RLQQ46AKP
Target Activities
30 Activities
Items per page:
1 – 10 of 30
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