vinorelbine
A vinca alkaloid related to VINBLASTINE that is used as a first-line treatment for NON-SMALL CELL LUNG CANCER, or for advanced or metastatic BREAST CANCER refractory to treatment with ANTHRACYCLINES.
Ligand Summary
UNII: Q6C979R91Y
PubChem: 16051941
PubChem: 5311497
ChEMBL: CHEMBL538943
ChEMBL: CHEMBL553025
DrugCentral: 2827
LyCHI: XCK2T8GMAGSV
Target Activities
CYP3A4
Cytochrome P450 3A4
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IC50 | 6 | None, None:None:None | ||||
TUBB
Tubulin beta chain
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TUBB1
Tubulin beta-1 chain
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TUBB2A
Tubulin beta-2A chain
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TUBB2B
Tubulin beta-2B chain
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TUBB3
Tubulin beta-3 chain
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TUBB4A
Tubulin beta-4A chain
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TUBB4B
Tubulin beta-4B chain
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TUBB6
Tubulin beta-6 chain
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TUBB8
Tubulin beta-8 chain
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