varenicline
Ligand Summary
A benzazepine derivative that functions as an ALPHA4-BETA2 NICOTINIC RECEPTOR partial agonist. It is used for SMOKING CESSATION.
UNII: W6HS99O8ZO
PubChem: 170361
PubChem: 5310966
Guide to Pharmacology: 5459
ChEMBL: CHEMBL1396
DrugCentral: 2808
LyCHI: 3TAPHRAR5C42
Target Activities
4 Activities
Items per page:
1 – 4 of 4
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | AGONIST | |||||
Ki | AGONIST | |||||
Ki | ||||||