ulipristal
Ligand Summary
Ulipristal acetate is a selective progesterone receptor modulator with antagonistic and partial agonistic effects (a progesterone agonist/antagonist) at the progesterone receptor. It binds the human progesterone receptor and prevents progesterone from occupying its receptor. The likely primary mechanism of action of ulipristal acetate for emergency contraception is inhibition or delay of ovulation.
UNII: YF7V70N02B
PubChem: 13559281
PubChem: 130904
Guide to Pharmacology: 7460
ChEMBL: CHEMBL2103846
ChEMBL: CHEMBL260538
DrugCentral: 4166
LyCHI: SQMHQGH31URQ
Target Activities
4 Activities
Items per page:
10
1 – 4 of 4
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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EC50 | ||||||
IC50 | ||||||
IC50 | ||||||
IC50 | ANTAGONIST | |||||