tiagabine
Ligand Summary
The precise mechanism by which tiagabine exerts its antiseizure effect is unknown, although it is believed to be related to its ability to block GABA uptake into presynaptic neurons, permitting more GABA to be available for receptor binding on the surfaces of post-synaptic cells.
UNII: Z80I64HMNP
PubChem: 60648
PubChem: 91274
Guide to Pharmacology: 4818
ChEMBL: CHEMBL1027
ChEMBL: CHEMBL1695
DrugCentral: 2648
LyCHI: KWXTL21QA8XP
Target Activities
11 Activities
Items per page:
1 – 10 of 11
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