tezacaftor
Ligand Summary
Tezacaftor facilitates the cellular processing and trafficking of normal and select mutant forms of CFTR (including F508del-CFTR) to increase the amount of mature CFTR protein delivered to the cell surface.
UNII: 8RW88Y506K
PubChem: 46199646
Guide to Pharmacology: 10199
ChEMBL: CHEMBL3544914
DrugCentral: 5276
LyCHI: J4BJ26SGQ4NJ
Target Activities
4 Activities
Items per page:
1 – 4 of 4
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EC50 | PHARMACOLOGICAL CHAPERONE | |||||