tazarotene
a topical acetylenic retinoid; a topical kerytolytic
Ligand Summary
UNII: 81BDR9Y8PS
PubChem: 5381
Guide to Pharmacology: 6952
ChEMBL: CHEMBL1657
DrugCentral: 2571
LyCHI: PVZSWAXQMF34
Target Activities
RARA
Retinoic acid receptor alpha
3 Activities
Items per page:
1 – 3 of 3
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
EC50 | 7.2 | |||||
EC50 | 7.2 | Bioorg. Med. Chem. Lett., (2009) 19:2:489 | ||||
EC50 | 7.2 | AGONIST | ||||
RARB
Retinoic acid receptor beta
3 Activities
Items per page:
1 – 3 of 3
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
EC50 | 9.1 | |||||
EC50 | 9.1 | Bioorg. Med. Chem. Lett., (2009) 19:2:489 | ||||
EC50 | 9.1 | AGONIST | ||||
RARG
Retinoic acid receptor gamma
3 Activities
Items per page:
1 – 3 of 3
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
EC50 | 7.4 | |||||
EC50 | 7.4 | Bioorg. Med. Chem. Lett., (2009) 19:2:489 | ||||
EC50 | 7.4 | AGONIST | ||||