tamoxifen
Ligand Summary
One of the SELECTIVE ESTROGEN RECEPTOR MODULATORS with tissue-specific activities. Tamoxifen acts as an anti-estrogen (inhibiting agent) in the mammary tissue, but as an estrogen (stimulating agent) in cholesterol metabolism, bone density, and cell proliferation in the ENDOMETRIUM.
UNII: 094ZI81Y45
PubChem: 2733526
PubChem: 139148739
Guide to Pharmacology: 1016
ChEMBL: CHEMBL83
ChEMBL: CHEMBL786
DrugCentral: 2561
LyCHI: 77VBQQV883JS
Target Activities
42 Activities
Items per page:
1 – 10 of 42
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
- | ||||||
- | ||||||
IC50 | ||||||
Ki | ||||||
Ki | ||||||
IC50 | ||||||
Ki | ||||||