sulindac
Ligand Summary
A sulfinylindene derivative prodrug whose sulfinyl moiety is converted in vivo to an active NSAID analgesic. Specifically, the prodrug is converted by liver enzymes to a sulfide which is excreted in the bile and then reabsorbed from the intestine. This helps to maintain constant blood levels with reduced gastrointestinal side effects.
UNII: 184SNS8VUH
PubChem: 1548887
Guide to Pharmacology: 5425
ChEMBL: CHEMBL15770
DrugCentral: 2534
LyCHI: CLRLMAWF3NSM
Target Activities
8 Activities
Items per page:
1 – 8 of 8
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