setmelanotide
Ligand Summary
Setmelanotide is an 8 amino acid cyclic peptide analog of endogenous melanocortin peptide alpha-MSH (alpha-melanocyte stimulating hormone). It is a melanocortin 4 (MC4) receptor agonist, with 20-fold less activity at the melanocortin 3 (MC3) and melanocortin 1 (MC1) receptors.
PubChem: 11993702
ChEMBL: CHEMBL3301624
DrugCentral: 5416
LyCHI: VNK5R8586QRH
Target Activities
2 Activities
Items per page:
1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Kd | AGONIST | |||||
Ki | AGONIST | |||||