Romidepsin
Ligand Summary
Target Activities
HDAC1
Histone deacetylase 1
4 Activities
Items per page:
1 – 4 of 4
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 8.8 | J Med Chem, (2020) 63:1:23 | ||||
IC50 | 8.62 | MedChemComm, (2019) 10:4:538 | ||||
IC50 | 7.44 | Eur J Med Chem, (2019) 183:None:111691 | ||||
IC50 | 7.44 | Eur J Med Chem, (2018) 158:None:620 | ||||
HDAC2
Histone deacetylase 2
3 Activities
HDAC6
Histone deacetylase 6
2 Activities
Items per page:
1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 8.04 | MedChemComm, (2019) 10:4:538 | ||||
IC50 | 6.1 | J Med Chem, (2020) 63:1:23 | ||||
HDAC4
Histone deacetylase 4
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 6.29 | Eur J Med Chem, (2018) 158:None:620 | ||||