olmesartan medoxomil
Ligand Summary
Olmesartan blocks the vasoconstrictor effects of angiotensin II by selectively blocking the binding of angiotensin II to the AT1 receptor in vascular smooth muscle.
UNII: 6M97XTV3HD
PubChem: 130881
Guide to Pharmacology: 591
ChEMBL: CHEMBL1200692
DrugCentral: 1985
LyCHI: KUVPWHRXXN1N
Target Activities
AGTR1
Type-1 angiotensin II receptor
2 Activities
Items per page:
1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
- | 8.1 | |||||
IC50 | 8.1 | ANTAGONIST | ||||