You are using an outdated browser. Please upgrade your browser to improve your experience.

oliceridine

Ligand Summary
Ligand Structure
Rendered image for the query structure
Description
Oliceridine is a full opioid agonist and is relatively selective for the mu-opioid receptor. The principal therapeutic action of oliceridine is analgesia. Like all full opioid agonists, there is no ceiling effect to analgesia for oliceridine. Clinically, dosage is titrated to provide adequate analgesia and may be limited by adverse reactions, including respiratory, and CNS depression. The precise mechanism of the analgesic action is unknown. However, specific CNS opioid receptors for endogenous compounds with opioid-like activity have been identified throughout the brain and spinal cord and are thought to play a role in the analgesic effects of this drug.
Synonyms & Links
DrugCentral: 5406
LyCHI:  SXKPY5R41KAR


Target Activities