octreotide
Ligand Summary
A potent, long-acting synthetic SOMATOSTATIN octapeptide analog that inhibits secretion of GROWTH HORMONE and is used to treat hormone-secreting tumors; DIABETES MELLITUS; HYPOTENSION, ORTHOSTATIC; HYPERINSULINISM; hypergastrinemia; and small bowel fistula.
UNII: RWM8CCW8GP
PubChem: 448601
ChEMBL: CHEMBL1680
DrugCentral: 1980
LyCHI: 8GQHYX4RF41G
Target Activities
5 Activities
Items per page:
10
1 – 5 of 5
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
EC50 | AGONIST | |||||
Ki | AGONIST | |||||
IC50 | AGONIST | |||||
Ki | AGONIST | |||||
Ki | AGONIST | |||||