nitroxoline
Ligand Summary
UNII: A8M33244M6
PubChem: 19910
ChEMBL: CHEMBL1454910
DrugCentral: 1954
LyCHI: QJHCLT7QDGF4
Target Activities
METAP2
Methionine aminopeptidase 2
3 Activities
Items per page:
1 – 3 of 3
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 7.26 | ACS Med. Chem. Lett., (2013) 4:8:699 | ||||
IC50 | 7.26 | J Med Chem, (2019) 62:10:5025 | ||||
IC50 | 7.26 | |||||
BRD4
Bromodomain-containing protein 4
3 Activities
Items per page:
1 – 3 of 3
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 6.01 | Eur J Med Chem, (2019) 163:None:281 | ||||
IC50 | 6.01 | Eur J Med Chem, (2019) 163:None:281 | ||||
IC50 | 6.01 | |||||
HSP90AA1
Heat shock protein HSP 90-alpha
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
AC50 | 6 | None, None:None:None | ||||
PTGS2
Prostaglandin G/H synthase 2
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 6 | J. Med. Chem., (2013) 56:21:8377 | ||||