laropiprant
a potent orally active human prostaglandin D(2) receptor 1 antagonist
Ligand Summary
Target Activities
PTGDR
Prostaglandin D2 receptor
6 Activities
Items per page:
1 – 6 of 6
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 10.52 | J. Med. Chem., (2007) 50:4:794 | ||||
IC50 | 10.05 | J. Med. Chem., (2007) 50:4:794 | ||||
Ki | 9.24 | J. Med. Chem., (2007) 50:4:794 | ||||
IC50 | 8.85 | J. Med. Chem., (2007) 50:4:794 | ||||
IC50 | 8.4 | J. Med. Chem., (2007) 50:4:794 | ||||
Kd | 10.52 | ANTAGONIST | ||||