halothane
Ligand Summary
A nonflammable, halogenated, hydrocarbon anesthetic that provides relatively rapid induction with little or no excitement. Analgesia may not be adequate. NITROUS OXIDE is often given concomitantly. Because halothane may not produce sufficient muscle relaxation, supplemental neuromuscular blocking agents may be required. (From AMA Drug Evaluations Annual, 1994, p178)
UNII: UQT9G45D1P
PubChem: 3562
Guide to Pharmacology: 2401
ChEMBL: CHEMBL931
DrugCentral: 1356
LyCHI: 7WYG58Z3XPYY
Target Activities
KCNK3
Potassium channel subfamily K member 3
2 Activities
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EC50 | 3 | |||||
OPENER | ||||||
KCNK5
Potassium channel subfamily K member 5
1 Activities
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3.7 | ||||||
KCNB1
Potassium voltage-gated channel subfamily B member 1
1 Activities
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3.5 | ||||||
GABRP
Gamma-aminobutyric acid receptor subunit pi
1 Activities
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GABRD
Gamma-aminobutyric acid receptor subunit delta
1 Activities
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GABRA1
Gamma-aminobutyric acid receptor subunit alpha-1
1 Activities
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GABRB1
Gamma-aminobutyric acid receptor subunit beta-1
1 Activities
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GABRG2
Gamma-aminobutyric acid receptor subunit gamma-2
1 Activities
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GABRB3
Gamma-aminobutyric acid receptor subunit beta-3
1 Activities
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GABRA5
Gamma-aminobutyric acid receptor subunit alpha-5
1 Activities
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GABRA3
Gamma-aminobutyric acid receptor subunit alpha-3
1 Activities
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GABRA2
Gamma-aminobutyric acid receptor subunit alpha-2
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GABRB2
Gamma-aminobutyric acid receptor subunit beta-2
1 Activities
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GABRA4
Gamma-aminobutyric acid receptor subunit alpha-4
1 Activities
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GABRE
Gamma-aminobutyric acid receptor subunit epsilon
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GABRA6
Gamma-aminobutyric acid receptor subunit alpha-6
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GABRG1
Gamma-aminobutyric acid receptor subunit gamma-1
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GABRG3
Gamma-aminobutyric acid receptor subunit gamma-3
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GABRQ
Gamma-aminobutyric acid receptor subunit theta
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KCNK2
Potassium channel subfamily K member 2
1 Activities
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OPENER | ||||||
KCNK9
Potassium channel subfamily K member 9
1 Activities
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KCNK10
Potassium channel subfamily K member 10
1 Activities
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KCNK18
Potassium channel subfamily K member 18
1 Activities
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GLRA1
Glycine receptor subunit alpha-1
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GLRB
Glycine receptor subunit beta
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