eslicarbazepine acetate
Eslicarbazepine acetate is extensively converted to eslicarbazepine, which is considered to be responsible for therapeutic effects in humans. The precise mechanism(s) by which eslicarbazepine exerts anticonvulsant activity is unknown but is thought to involve inhibition of voltage-gated sodium channels.
Ligand Summary
Target Activities
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SCN1A
Sodium channel protein type 1 subunit alpha
1 Activities
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BLOCKER | ||||||
SCN4A
Sodium channel protein type 4 subunit alpha
1 Activities
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BLOCKER | ||||||
SCN7A
Sodium channel protein type 7 subunit alpha
1 Activities
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BLOCKER | ||||||
SCN5A
Sodium channel protein type 5 subunit alpha
1 Activities
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BLOCKER | ||||||
SCN9A
Sodium channel protein type 9 subunit alpha
1 Activities
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BLOCKER | ||||||
SCN2A
Sodium channel protein type 2 subunit alpha
1 Activities
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BLOCKER | ||||||
SCN3A
Sodium channel protein type 3 subunit alpha
1 Activities
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BLOCKER | ||||||
SCN11A
Sodium channel protein type 11 subunit alpha
1 Activities
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BLOCKER | ||||||
SCN8A
Sodium channel protein type 8 subunit alpha
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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BLOCKER | ||||||
SCN10A
Sodium channel protein type 10 subunit alpha
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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BLOCKER | ||||||