eplerenone
Ligand Summary
A spironolactone derivative and selective ALDOSTERONE RECEPTOR antagonist that is used in the management of HYPERTENSION and CONGESTIVE HEART FAILURE, post-MYOCARDIAL INFARCTION.
UNII: 6995V82D0B
PubChem: 443872
Guide to Pharmacology: 2876
ChEMBL: CHEMBL1095097
DrugCentral: 1032
LyCHI: KDJTD4QDC3Y7
Target Activities
4 Activities
Items per page:
10
1 – 4 of 4
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Ki | ||||||
IC50 | ||||||
EC50 | ||||||
IC50 | ANTAGONIST | |||||