cimetidine
Ligand Summary
A histamine congener, it competitively inhibits HISTAMINE binding to HISTAMINE H2 RECEPTORS. Cimetidine has a range of pharmacological actions. It inhibits GASTRIC ACID secretion, as well as PEPSIN and GASTRIN output.
UNII: 80061L1WGD
PubChem: 2756
Guide to Pharmacology: 1231
ChEMBL: CHEMBL30
DrugCentral: 645
LyCHI: 2HM79A95BD25
Target Activities
8 Activities
Items per page:
1 – 8 of 8
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Ki | ||||||
- | ||||||
Ki | ||||||
Ki | ||||||
Ki | ||||||
Ki | ||||||
Ki | ||||||
Kd | ANTAGONIST | |||||