Chidamide
Ligand Summary
Target Activities
HDAC1
Histone deacetylase 1
6 Activities
Items per page:
1 – 6 of 6
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 7.02 | Eur J Med Chem, (2019) 183:None:111691 | ||||
IC50 | 6.8 | Bioorg Med Chem Lett, (2020) 30:8:127036 | ||||
IC50 | 6.72 | Eur J Med Chem, (2019) 173:None:185 | ||||
IC50 | 6.72 | Eur J Med Chem, (2019) 176:None:195 | ||||
IC50 | 6.27 | Eur J Med Chem, (2018) 143:None:320 | ||||
IC50 | 6.06 | Bioorg Med Chem Lett, (2017) 27:14:3162 | ||||
HDAC2
Histone deacetylase 2
4 Activities
Items per page:
1 – 4 of 4
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 6.8 | Eur J Med Chem, (2019) 183:None:111691 | ||||
IC50 | 6.51 | Eur J Med Chem, (2019) 173:None:185 | ||||
IC50 | 6.51 | Eur J Med Chem, (2019) 176:None:195 | ||||
IC50 | 6.43 | Eur J Med Chem, (2018) 143:None:320 | ||||
HDAC3
Histone deacetylase 3
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 7.17 | Eur J Med Chem, (2019) 183:None:111691 | ||||
HDAC10
Histone deacetylase 10
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 7.11 | Eur J Med Chem, (2019) 183:None:111691 | ||||