brigatinib
Ligand Summary
Name: brigatinib
PubChem: 57390074
Guide to Pharmacology: 7741
ChEMBL: CHEMBL3397300
LyCHI: NSL4GK65GM2W
Target Activities
ALK
ALK tyrosine kinase receptor
3 Activities
IGF1R
Insulin-like growth factor 1 receptor
2 Activities
EGFR
Epidermal growth factor receptor
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 6.89 | |||||
INSR
Insulin receptor
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 6.71 | |||||
ROS1
Proto-oncogene tyrosine-protein kinase ROS
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 8.72 | Eur. J. Med. Chem., (2015) 90:None:195 | ||||