R547
Ligand Summary
Name: R547
PubChem: 6918852
Guide to Pharmacology: 5707
ChEMBL: CHEMBL384304
LyCHI: ZZ7KN7848XXD
Target Activities
CDK2
Cyclin-dependent kinase 2
5 Activities
Items per page:
1 – 5 of 5
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 9.28 | |||||
Ki | 8.52 | |||||
Kd | 9.28 | Nat. Biotechnol., (2011) 29:11:1046 | ||||
Ki | 8.52 | J. Med. Chem., (2006) 49:22:6549 | ||||
Kd | 8.3 | Science, (2017) 358:6367:None | ||||
CDK4
Cyclin-dependent kinase 4
3 Activities
CDK1
Cyclin-dependent kinase 1
2 Activities
CDK9
Cyclin-dependent kinase 9
2 Activities
CDK5
Cyclin-dependent-like kinase 5
2 Activities
DYRK1A
Dual specificity tyrosine-phosphorylation-regulated kinase 1A
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 7.64 | Nat. Biotechnol., (2011) 29:11:1046 | ||||
CDK7
Cyclin-dependent kinase 7
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 9.24 | Nat. Biotechnol., (2011) 29:11:1046 | ||||
CLK3
Dual specificity protein kinase CLK3
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 7.89 | Nat. Biotechnol., (2011) 29:11:1046 | ||||
CDK3
Cyclin-dependent kinase 3
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 8.49 | Nat. Biotechnol., (2011) 29:11:1046 | ||||
MAPK15
Mitogen-activated protein kinase 15
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 7.75 | Science, (2017) 358:6367:None | ||||
CDK18
Cyclin-dependent kinase 18
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 7.7 | Nat. Biotechnol., (2011) 29:11:1046 | ||||
CDK17
Cyclin-dependent kinase 17
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 9.07 | Nat. Biotechnol., (2011) 29:11:1046 | ||||
CDK15
Cyclin-dependent kinase 15
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 8.14 | Nat. Biotechnol., (2011) 29:11:1046 | ||||
CDK14
Cyclin-dependent kinase 14
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 7.96 | Nat. Biotechnol., (2011) 29:11:1046 | ||||
MAK
Serine/threonine-protein kinase MAK
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 7.96 | Nat. Biotechnol., (2011) 29:11:1046 | ||||
ICK
Serine/threonine-protein kinase ICK
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 8.66 | Nat. Biotechnol., (2011) 29:11:1046 | ||||
CDK16
Cyclin-dependent kinase 16
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 9.27 | Nat. Biotechnol., (2011) 29:11:1046 | ||||