fasiglifam
Ligand Summary
Name: fasiglifam
PubChem: 24857286
PubChem: 46869922
Guide to Pharmacology: 6484
ChEMBL: CHEMBL1829174
ChEMBL: CHEMBL2047159
LyCHI: ZZ2744RC8RJV
Target Activities
FFAR1
Free fatty acid receptor 1
30 Activities
Items per page:
1 – 10 of 30
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
- | 7.1 | |||||
EC50 | 8.72 | ACS Med Chem Lett, (2016) 7:12:1134 | ||||
EC50 | 8.03 | J. Med. Chem., (2016) 59:10:4849 | ||||
EC50 | 7.85 | J. Med. Chem., (2011) 54:19:6691 | ||||
EC50 | 7.85 | ACS Med. Chem. Lett., (2010) 1:6:290 | ||||
EC50 | 7.85 | ACS Med Chem Lett, (2017) 8:12:1336 | ||||
EC50 | 7.85 | Eur J Med Chem, (2018) 159:None:267 | ||||
EC50 | 7.8 | J. Med. Chem., (2012) 55:8:3960 | ||||
EC50 | 7.57 | J Med Chem, (2017) 60:7:2697 | ||||
EC50 | 7.56 | Eur. J. Med. Chem., (2016) 116:None:46 | ||||