Pharos : Ligand Details - ZTH9MPJPQ1FS

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Ligand Summary

Ligand Structure

Rendered image for the query structure

Synonyms & Links

Name: LG100754

PubChem: 6442223

Guide to Pharmacology: 2814

ChEMBL: CHEMBL109581

LyCHI: ZTH9MPJPQ1FS

Target Activities

RXRA

Tclin

Retinoic acid receptor RXR-alpha

3 Activities

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1 – 3 of 3

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
-	8.5			11463859

EC50	8.7		J. Med. Chem., (1996) 39:17:3229	8765503

Ki	8.1		J. Med. Chem., (1996) 39:17:3229	8765503

RXRB

Tclin

Retinoic acid receptor RXR-beta

3 Activities

Items per page:

1 – 3 of 3

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
	8			11463859 11877384 8837780

Ki	8.05		J. Med. Chem., (1996) 39:17:3229	8765503

EC50	7.89		J. Med. Chem., (1996) 39:17:3229	8765503

RXRG

Tclin

Retinoic acid receptor RXR-gamma

2 Activities

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1 – 2 of 2

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
EC50	8.4		J. Med. Chem., (1996) 39:17:3229	8765503

Ki	7.85		J. Med. Chem., (1996) 39:17:3229	8765503

RARB

Tclin

Retinoic acid receptor beta

1 Activities

Items per page:

1 – 1 of 1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
EC50	8		J. Med. Chem., (1996) 39:17:3229	8765503

RARA

Tclin

Retinoic acid receptor alpha

1 Activities

Items per page:

1 – 1 of 1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
EC50	8.4		J. Med. Chem., (1996) 39:17:3229	8765503