PB28
Ligand Summary
Name: PB28
PubChem: 10474335
PubChem: 10361439
Guide to Pharmacology: 6681
ChEMBL: CHEMBL53325
ChEMBL: CHEMBL322275
LyCHI: ZPSUZG3BHZSL
Target Activities
SIGMAR1
Sigma non-opioid intracellular receptor 1
7 Activities
Items per page:
1 – 7 of 7
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Ki | 8.7 | Nature, (2020) None:None:None | ||||
Ki | 8.28 | J. Med. Chem., (1996) 39:1:176 | ||||
Ki | 7.89 | Bioorg. Med. Chem., (2014) 22:1:221 | ||||
Ki | 7.89 | J. Med. Chem., (2014) 57:10:4239 | ||||
Ki | 7.87 | J. Med. Chem., (2004) 47:9:2308 | ||||
Ki | 7.87 | Eur J Med Chem, (2018) 147:None:227 | ||||
IC50 | 6.7 | J. Med. Chem., (1995) 38:6:942 | ||||
TMEM97
Sigma intracellular receptor 2
3 Activities
KCNH2
Potassium voltage-gated channel subfamily H member 2
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Ki | 6 | Nature, (2020) None:None:None | ||||
ABCB1
Multidrug resistance protein 1
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
EC50 | 6.26 | Bioorg. Med. Chem., (2008) 16:1:362 | ||||