Pharos : Ligand Details - ZMF3WFHQ7CDT

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Ligand Summary

Ligand Structure

chemical structure image

Synonyms & Links

Name: Valethamate Bromide

PubChem: 7010

ChEMBL: CHEMBL2107687

LyCHI: ZMF3WFHQ7CDT

Target Activities

CHRM3

Tclin

Muscarinic acetylcholine receptor M3

2 Activities

Items per page:

1 – 2 of 2

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	7.58		None, None:None:None

Ki	8.25		None, None:None:None

CHRM1

Tclin

Muscarinic acetylcholine receptor M1

2 Activities

Items per page:

1 – 2 of 2

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	7.92		None, None:None:None

Ki	8.56		None, None:None:None

CHRM2

Tclin

Muscarinic acetylcholine receptor M2

2 Activities

Items per page:

1 – 2 of 2

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	7.26		None, None:None:None

Ki	7.72		None, None:None:None

CHRM4

Tclin

Muscarinic acetylcholine receptor M4

2 Activities

Items per page:

1 – 2 of 2

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	7.58		None, None:None:None

Ki	8.44		None, None:None:None

CHRM5

Tclin

Muscarinic acetylcholine receptor M5

2 Activities

Items per page:

1 – 2 of 2

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	7.47		None, None:None:None

Ki	7.62		None, None:None:None

SIGMAR1

Tclin

Sigma non-opioid intracellular receptor 1

2 Activities

Items per page:

1 – 2 of 2

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	6.32		None, None:None:None

Ki	6.7		None, None:None:None

CYP2D6

Tclin

Cytochrome P450 2D6

1 Activities

Items per page:

1 – 1 of 1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	6.61		None, None:None:None