Valethamate Bromide
Ligand Summary
Target Activities
CHRM3
Muscarinic acetylcholine receptor M3
2 Activities
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1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 8.25 | None, None:None:None | ||||
IC50 | 7.58 | None, None:None:None | ||||
CHRM4
Muscarinic acetylcholine receptor M4
2 Activities
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1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 8.44 | None, None:None:None | ||||
IC50 | 7.58 | None, None:None:None | ||||
CHRM1
Muscarinic acetylcholine receptor M1
2 Activities
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1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 8.56 | None, None:None:None | ||||
IC50 | 7.92 | None, None:None:None | ||||
SIGMAR1
Sigma non-opioid intracellular receptor 1
2 Activities
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1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 6.7 | None, None:None:None | ||||
IC50 | 6.32 | None, None:None:None | ||||
CHRM5
Muscarinic acetylcholine receptor M5
2 Activities
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1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 7.62 | None, None:None:None | ||||
IC50 | 7.47 | None, None:None:None | ||||
CHRM2
Muscarinic acetylcholine receptor M2
2 Activities
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1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 7.72 | None, None:None:None | ||||
IC50 | 7.26 | None, None:None:None | ||||
CYP2D6
Cytochrome P450 2D6
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 6.61 | None, None:None:None | ||||