Bromosporine
Ligand Summary
Target Activities
BRD4
Bromodomain-containing protein 4
5 Activities
Items per page:
1 – 5 of 5
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Kd | 7.38 | J Med Chem, (2020) 63:6:3227 | ||||
IC50 | 7.08 | Science Advances, (2016) None:10:e1600760 | ||||
IC50 | 6.93 | Science Advances, (2016) None:10:e1600760 | ||||
IC50 | 6.51 | Science Advances, (2016) None:10:e1600760 | ||||
IC50 | 6.33 | Science Advances, (2016) None:10:e1600760 | ||||
CECR2
Cat eye syndrome critical region protein 2
5 Activities
Items per page:
1 – 5 of 5
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 8.1 | Science Advances, (2016) None:10:e1600760 | ||||
IC50 | 8.03 | Science Advances, (2016) None:10:e1600760 | ||||
Kd | 8 | J Med Chem, (2020) 63:10:5212 | ||||
IC50 | 7.32 | Science Advances, (2016) None:10:e1600760 | ||||
IC50 | 7.1 | Science Advances, (2016) None:10:e1600760 | ||||
BRD9
Bromodomain-containing protein 9
5 Activities
Items per page:
1 – 5 of 5
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 7.33 | Science Advances, (2016) None:10:e1600760 | ||||
Kd | 6.94 | J Med Chem, (2020) 63:6:3227 | ||||
IC50 | 6.8 | Bioorg Med Chem, (2019) 27:7:1391 | ||||
IC50 | 6.52 | Science Advances, (2016) None:10:e1600760 | ||||
IC50 | 6.15 | Science Advances, (2016) None:10:e1600760 | ||||
BRDT
Bromodomain testis-specific protein
2 Activities
BRD2
Bromodomain-containing protein 2
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Kd | 7.3 | Science Advances, (2016) None:10:e1600760 | ||||
BRD7
Bromodomain-containing protein 7
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Kd | 6.41 | J Med Chem, (2020) 63:6:3227 | ||||
BRPF1
Peregrin
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 6.85 | Science Advances, (2016) None:10:e1600760 | ||||
TAF1
Transcription initiation factor TFIID subunit 1
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 7.78 | Science Advances, (2016) None:10:e1600760 | ||||