CHEMBL4449894
Ligand Summary
Name: N-(4-Bromo-3-(((S)-3-methylpyrrolidin-1-yl)sulfonyl)phenyl)-2-((S)-4-cyclopropyl-4-methyl-2,5-dioxoimidazolidin-1-yl)acetamide
PubChem: 155521254
ChEMBL: CHEMBL4449894
LyCHI: YW97GNT7VUXC
Target Activities
CECR2
Cat eye syndrome critical region protein 2
3 Activities
ATAD2
ATPase family AAA domain-containing protein 2
2 Activities
KAT2A
Histone acetyltransferase KAT2A
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 6.6 | J Med Chem, (2020) 63:10:5212 | ||||
BRD1
Bromodomain-containing protein 1
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 6.9 | J Med Chem, (2020) 63:10:5212 | ||||
ATAD2B
ATPase family AAA domain-containing protein 2B
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 7.7 | J Med Chem, (2020) 63:10:5212 | ||||
TAF1
Transcription initiation factor TFIID subunit 1
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 7.8 | J Med Chem, (2020) 63:10:5212 | ||||
TAF1L
Transcription initiation factor TFIID subunit 1-like
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 7.6 | J Med Chem, (2020) 63:10:5212 | ||||
BAZ2A
Bromodomain adjacent to zinc finger domain protein 2A
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 7.8 | J Med Chem, (2020) 63:10:5212 | ||||
BRPF3
Bromodomain and PHD finger-containing protein 3
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 6.9 | J Med Chem, (2020) 63:10:5212 | ||||