Bardoxolone methyl
Ligand Summary
Name: Bardoxolone methyl
PubChem: 400769
Guide to Pharmacology: 3443
ChEMBL: CHEMBL1762621
LyCHI: YSAB3DBC197N
Target Activities
PPARG
Peroxisome proliferator-activated receptor gamma
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 6.9 | |||||
NFE2L2
Nuclear factor erythroid 2-related factor 2
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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EC50 | 7.22 | J Nat Prod, (2017) 80:8:2276 | ||||