2-APB
Ligand Summary
Name: 2-APB
PubChem: 1598
Guide to Pharmacology: 2433
ChEMBL: CHEMBL169233
LyCHI: XJS2H8DY719A
Target Activities
TRPM2
Transient receptor potential cation channel subfamily M member 2
3 Activities
TRPC3
Short transient receptor potential channel 3
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 5 | |||||
TRPC5
Short transient receptor potential channel 5
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 4.7 | |||||
TRPM3
Transient receptor potential cation channel subfamily M member 3
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
- | 4 | |||||
TRPM7
Transient receptor potential cation channel subfamily M member 7
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 3.75 | |||||
TRPV2
Transient receptor potential cation channel subfamily V member 2
1 Activities
TRPV3
Transient receptor potential cation channel subfamily V member 3
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
EC50 | 4.6 | |||||