IKK-2 inhibitor IV
Ligand Summary
Name: IKK-2 inhibitor IV
PubChem: 9903786
Guide to Pharmacology: 5986
ChEMBL: CHEMBL257167
LyCHI: XBS6877PWDJF
Target Activities
IKBKB
Inhibitor of nuclear factor kappa-B kinase subunit beta
5 Activities
Items per page:
1 – 5 of 5
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 7.75 | |||||
IC50 | 7.75 | J. Nat. Prod., (2008) 71:1:106 | ||||
IC50 | 7.75 | Bioorg. Med. Chem., (2009) 17:7:2759 | ||||
IC50 | 7.71 | J. Med. Chem., (2008) 51:24:7898 | ||||
IC50 | 7.7 | Bioorg. Med. Chem. Lett., (2011) 21:8:2255 | ||||