SAR407899
Ligand Summary
Name: SAR407899
PubChem: 15604510
Guide to Pharmacology: 8910
ChEMBL: CHEMBL1667969
LyCHI: X9K65KQMYCT6
Target Activities
ROCK2
Rho-associated protein kinase 2
4 Activities
ROCK1
Rho-associated protein kinase 1
2 Activities
PRKCD
Protein kinase C delta type
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 7.68 | Science, (2017) 358:6367:None | ||||
AAK1
AP2-associated protein kinase 1
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 7.92 | Science, (2017) 358:6367:None | ||||
PRKACA
cAMP-dependent protein kinase catalytic subunit alpha
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 7.89 | Science, (2017) 358:6367:None | ||||
PRKG1
cGMP-dependent protein kinase 1
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 8.4 | Science, (2017) 358:6367:None | ||||
CDC42BPA
Serine/threonine-protein kinase MRCK alpha
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 8 | Science, (2017) 358:6367:None | ||||
BMP2K
BMP-2-inducible protein kinase
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 7.89 | Science, (2017) 358:6367:None | ||||
PKN2
Serine/threonine-protein kinase N2
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 8.1 | Science, (2017) 358:6367:None | ||||
Q6ZSR9
Uncharacterized protein FLJ45252
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 7.89 | Science, (2017) 358:6367:None | ||||
CDC42BPB
Serine/threonine-protein kinase MRCK beta
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 7.8 | Science, (2017) 358:6367:None | ||||
PKN1
Serine/threonine-protein kinase N1
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 7.72 | Science, (2017) 358:6367:None | ||||