ethylisopropylamiloride
Ligand Summary
Name: ethylisopropylamiloride
PubChem: 1795
Guide to Pharmacology: 4186
ChEMBL: CHEMBL517986
LyCHI: X4A5Z4RDC2JZ
Target Activities
SLC9A5
Sodium/hydrogen exchanger 5
6 Activities
Items per page:
1 – 6 of 6
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 6.38 | None, (2014) None:None:None | ||||
Ki | 6.38 | None, (2013) None:None:None | ||||
IC50 | 6.38 | None, None:None:None | ||||
Ki | 6.38 | |||||
Ki | 6.38 | |||||
IC50 | 6.38 | |||||
ADRA2A
Alpha-2A adrenergic receptor
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
- | 1.8 | |||||
ASIC1
Acid-sensing ion channel 1
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 5 | |||||
PKD2L1
Polycystic kidney disease 2-like 1 protein
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 5 | |||||
SLC9A1
Sodium/hydrogen exchanger 1
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 6.1 | J. Biol. Chem., (2007) 282:27:19716 | ||||