CHEMBL129857
Ligand Summary
NCATS Inxight: Drugs: 9820526
Name: 1-(5-methoxy-2-(thiophen-2-yl)quinazolin-4-ylamino)-3-methyl-1H-pyrrole-2,5-dione
PubChem: 9820526
ChEMBL: CHEMBL129857
LyCHI: WD391N7NADVH
Target Activities
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10
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JUN
Transcription factor AP-1
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 8.1 | J. Med. Chem., (2014) 57:16:6930 | ||||
IKBKB
Inhibitor of nuclear factor kappa-B kinase subunit beta
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 8.1 | Bioorg. Med. Chem., (2009) 17:7:2759 | ||||
RELA
Transcription factor p65
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
EC50 | 6.42 | Bioorg. Med. Chem. Lett., (2009) 19:4:1191 | ||||