MK-5108
Ligand Summary
Name: MK-5108
PubChem: 24748204
Guide to Pharmacology: 8061
ChEMBL: CHEMBL3182444
LyCHI: VUNAPND3VJVB
Target Activities
AURKA
Aurora kinase A
2 Activities
AURKB
Aurora kinase B
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 7.85 | |||||
AURKC
Aurora kinase C
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 7.92 | |||||
JAK2
Tyrosine-protein kinase JAK2
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 7.6 | Science, (2017) 358:6367:None | ||||
IRAK3
Interleukin-1 receptor-associated kinase 3
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 7.62 | Science, (2017) 358:6367:None | ||||
BCR
Breakpoint cluster region protein
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 7.96 | Science, (2017) 358:6367:None | ||||
TNK1
Non-receptor tyrosine-protein kinase TNK1
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 8.22 | Science, (2017) 358:6367:None | ||||