ZD7288
Ligand Summary
Name: ZD7288
PubChem: 123984
PubChem: 123983
Guide to Pharmacology: 2359
ChEMBL: CHEMBL2052019
LyCHI: VH6GPWWYZ7F1
Target Activities
HCN1
Potassium/sodium hyperpolarization-activated cyclic nucleotide-gated channel 1
2 Activities
HCN4
Potassium/sodium hyperpolarization-activated cyclic nucleotide-gated channel 4
2 Activities
HCN2
Potassium/sodium hyperpolarization-activated cyclic nucleotide-gated channel 2
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 4.4 | |||||
HCN3
Potassium/sodium hyperpolarization-activated cyclic nucleotide-gated channel 3
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 4.5 | |||||