CHEMBL406027
Ligand Summary
Name: (4R)-4-[(1S,2S,7S,9R,10R,11S,14R,15R,16S)-9,16-dihydroxy-2,15-dimethyl-5-{N-methyl[3-({4-[(10S,11S,14R,15S,17R)-14-ethynyl-14-hydroxy-15-methyl-5-oxotetracyclo[8.7.0.0^{2,7}.0^{11,15}]heptadeca-1,6-dien-17-yl]phenyl}(methyl)amino)propane]sulfonamido}tetracyclo[8.7.0.0^{2,7}.0^{11,15}]heptadecan-14-yl]pentanoic acid
PubChem: 44396250
ChEMBL: CHEMBL406027
LyCHI: VG6U5S824J4K
Target Activities
NR3C1
Glucocorticoid receptor
3 Activities
ESR2
Estrogen receptor beta
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Ki | 7.41 | J. Med. Chem., (2004) 47:17:4213 | ||||
ESR1
Estrogen receptor
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Ki | 7.72 | J. Med. Chem., (2004) 47:17:4213 | ||||
PGR
Progesterone receptor
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Ki | 8.72 | J. Med. Chem., (2004) 47:17:4213 | ||||
AR
Androgen receptor
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Ki | 7.77 | J. Med. Chem., (2004) 47:17:4213 | ||||