CHEMBL4217292
Ligand Summary
Name: N-(1-((5-cyanopyridin-2-yl)methyl)-1H-pyrazol-3-yl)-2-(4-(1-(trifluoromethyl)cyclopropyl)phenyl)acetamide
PubChem: 118560618
ChEMBL: CHEMBL4217292
LyCHI: V9UHFG7CV7DH
Target Activities
CACNA1I
Voltage-dependent T-type calcium channel subunit alpha-1I
2 Activities
CACNA1H
Voltage-dependent T-type calcium channel subunit alpha-1H
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 7.75 | J Med Chem, (2017) 60:23:9769 | ||||
CACNA1C
Voltage-dependent L-type calcium channel subunit alpha-1C
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 5.62 | J Med Chem, (2017) 60:23:9769 | ||||
KCNH2
Potassium voltage-gated channel subfamily H member 2
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 5.26 | J Med Chem, (2017) 60:23:9769 | ||||
CACNA1G
Voltage-dependent T-type calcium channel subunit alpha-1G
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 8.19 | J Med Chem, (2017) 60:23:9769 | ||||