CHEMBL4081890
Ligand Summary
Name: 2-(3-([1,1'-biphenyl]-3-yl)-5-(cyclopropylmethyl)-4-(4-sulfamoylbenzyl)-1H-pyrazol-1-yl)thiazole-4-carboxylic acid
PubChem: 131955127
ChEMBL: CHEMBL4081890
LyCHI: TTWXD53L5ANK
Target Activities
LDHA
L-lactate dehydrogenase A chain
4 Activities
Items per page:
1 – 4 of 4
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 9.96 | J Med Chem, (2017) 60:22:9184 | ||||
IC50 | 7.5 | J Med Chem, (2017) 60:22:9184 | ||||
IC50 | 7.5 | J Med Chem, (2017) 60:22:9184 | ||||
EC50 | 6.77 | J Med Chem, (2017) 60:22:9184 | ||||
LDHB
L-lactate dehydrogenase B chain
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 7.57 | J Med Chem, (2017) 60:22:9184 | ||||