CHEMBL2206242
Ligand Summary
Name: (2R)-2-[(6-{[(5-Methylthiophen-2-yl)methyl]amino}-9-propyl-9H-purin-2-yl)amino]butan-1-ol
PubChem: 71463101
ChEMBL: CHEMBL2206242
LyCHI: TRZCWUTH3FRJ
Target Activities
CACNA1A
Voltage-dependent P/Q-type calcium channel subunit alpha-1A
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
EC50 | 5.06 | ACS Med. Chem. Lett., (2012) 3:12:985 | ||||
CACNA1B
Voltage-dependent N-type calcium channel subunit alpha-1B
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
EC50 | 5.14 | ACS Med. Chem. Lett., (2012) 3:12:985 | ||||