SP600125
Ligand Summary
Name: SP600125
PubChem: 8515
Guide to Pharmacology: 5273
ChEMBL: CHEMBL1725279
ChEMBL: CHEMBL7064
LyCHI: TQASGT2ZFMFV
Target Activities
MAPK10
Mitogen-activated protein kinase 10
3 Activities
MAPK8
Mitogen-activated protein kinase 8
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 7.4 | |||||
MAPK9
Mitogen-activated protein kinase 9
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 7.4 | |||||
FLT4
Vascular endothelial growth factor receptor 3
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 7.8 | None, None:None:None | ||||
CYP1A2
Cytochrome P450 1A2
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
AC50 | 7.8 | None, None:None:None | ||||
BMP2K
BMP-2-inducible protein kinase
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 7.6 | Nat. Biotechnol., (2005) 23:3:329 | ||||
MARK3
MAP/microtubule affinity-regulating kinase 3
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 8.4 | None, None:None:None | ||||
NTRK3
NT-3 growth factor receptor
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 8.1 | None, None:None:None | ||||
AURKB
Aurora kinase B
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 8 | None, None:None:None | ||||
CYP2D6
Cytochrome P450 2D6
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
AC50 | 6.4 | None, None:None:None | ||||