CHEMBL4635041
Ligand Summary
Name: (S)-3-(2-benzoyl-5-methyl-1,2,3,4-tetrahydroisoquinolin-7-yl)-3-(1-ethyl-4-methyl-1H-benzo[d][1,2,3]triazol-5-yl)propanoic acid
ChEMBL: CHEMBL4635041
LyCHI: TAN7AZ43KYJY
Target Activities
NFE2L2
Nuclear factor erythroid 2-related factor 2
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
EC50 | 6.57 | Bioorg Med Chem Lett, (2020) 30:4:126852 | ||||
KEAP1
Kelch-like ECH-associated protein 1
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 7.87 | Bioorg Med Chem Lett, (2020) 30:4:126852 | ||||