CHEMBL4643632
Ligand Summary
Name: 4-[(5-ethyl-11-methyl-6-oxo-pyrimido[4,5-b][1,4]benzodiazepin-2-yl)amino]-3-methoxy-N-(1-methyl-4-piperidyl)benzamide
ChEMBL: CHEMBL4643632
LyCHI: T584K3N5X3PZ
Target Activities
LRRK2
Leucine-rich repeat serine/threonine-protein kinase 2
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 7.85 | J Med Chem, (2020) 63:14:7817 | ||||
DCLK1
Serine/threonine-protein kinase DCLK1
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 8.7 | J Med Chem, (2020) 63:14:7817 | ||||
BRD4
Bromodomain-containing protein 4
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 6.28 | J Med Chem, (2020) 63:14:7817 | ||||