compound 13 [Chen <i>et al.</i>, 2016]
Ligand Summary
Name: compound 13 [Chen <i>et al.</i>, 2016]
PubChem: 121231410
Guide to Pharmacology: 9205
ChEMBL: CHEMBL4590355
LyCHI: SZBF1NWBUWHL
Target Activities
DOT1L
Histone-lysine N-methyltransferase, H3 lysine-79 specific
5 Activities
Items per page:
1 – 5 of 5
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Ki | 10.1 | |||||
Ki | 10.1 | ACS Med Chem Lett, (2016) 7:8:735 | ||||
IC50 | 9.4 | ACS Med Chem Lett, (2016) 7:8:735 | ||||
IC50 | 7.8 | ACS Med Chem Lett, (2016) 7:8:735 | ||||
IC50 | 6.47 | ACS Med Chem Lett, (2016) 7:8:735 | ||||